Azelastine (Nasal Route) Description and Brand Names (Azelastine Hydrochloride)

Azelastine nasal spray is available via prescription and over-the-counter for treating allergy symptoms. This antihistamine nasal spray effectively targets sneezing, itching, runny nose, watery eyes, and other allergy symptoms. However, there is more to this nasal spray than just its effectiveness. In this discussion, we will explore the description and brand names of azelastine, shedding light on its unique properties and potential benefits. So, let's dive into the world of azelastine and discover what makes it stand out among other allergy medications.

Key Takeaways

  • Astelin (azelastine) is an antihistamine nasal spray used to treat allergy symptoms.

  • It is indicated for the treatment of seasonal allergic rhinitis and vasomotor rhinitis.

  • Common side effects of Astelin include bitter taste, drowsiness, dizziness, and dry mouth.

  • Astelin should be used with caution in pregnant women and can interact with other medications that cause drowsiness.

Rhinolast
137mcg Spray

Prescription required. Product of UK/EU. Shipped from United Kingdom of Great Britain and Northern Ireland. Astelin is also marketed internationally under the name Rhinolast.


Generic equivalents for Astelin... What are generics?

Azelastine Hydrochloride
137mcg Spray

Prescription required. Product of India. Shipped from Mauritius.


To comply with Canadian International Pharmacy Association regulations you are permitted to order a 3-month supply or the closest package size available based on your personal prescription. read more

Medical Information

Here, we provide a brief overview of Astelin, related to its role in helping patients manage rhinitis symptoms.

Astelin Uses, Side Effects, and Dosage

The medical information pertaining to Astelin, including its uses, side effects, and dosage, provides valuable insights for healthcare professionals and patients seeking effective treatment options for nasal symptoms associated with allergies. Astelin is an antihistamine nasal spray used to treat symptoms such as sneezing, itching, and runny nose caused by seasonal allergic rhinitis and vasomotor rhinitis.

It can be used in adults, adolescents, and pediatric patients as young as 5 years old for seasonal allergies, and patients as young as 12 for chronic rhinitis. The recommended dose varies depending on the age and condition being treated, with one or two sprays per nostril one to two times daily being the usual recommendations.

Common side effects of Astelin include a bitter taste in the mouth, drowsiness, dizziness, nosebleeds, and dry mouth. It is important to prime the nasal spray before initial use and avoid spraying it into the eyes. Overall, the medical information provided about Astelin is crucial for healthcare professionals and patients to make informed decisions about its use.

Seasonal Allergic Rhinitis

Seasonal Allergic Rhinitis, also known as hay fever, is a common condition characterized by inflammation of the nasal passages due to an allergic reaction to airborne allergens such as pollen, mold spores, or pet dander. It is a bothersome condition that affects many individuals, causing symptoms such as sneezing, itching, runny nose, and nasal congestion.

These symptoms can significantly impact a person's quality of life, making it difficult to concentrate, sleep, or engage in daily activities. Fortunately, there are treatment options available to alleviate the symptoms of seasonal allergic rhinitis. One such option is Astelin, an antihistamine nasal spray that helps relieve symptoms like sneezing, itching, and runny nose caused by allergies. It is important to consult with a healthcare professional to determine the most appropriate treatment for your specific needs.

Azelastine May Relieve Nasal Congestion — Often the Most Bothersome Symptom For Many Allergy Sufferers

Nasal congestion, which is often the most bothersome symptom for individuals with allergies, has been proven to be effectively relieved by Astelin nasal spray. Astelin is an antihistamine nasal spray that can also help alleviate symptoms such as sneezing, itching, and a runny nose caused by allergies. By using Astelin nasal spray, individuals with allergies can experience relief from the uncomfortable symptoms of nasal congestion.

Drug Details

Now let's delve into the specific details about Astelin nasal spray. This antihistamine medication is indicated for the treatment of seasonal allergic rhinitis and vasomotor rhinitis. It helps relieve symptoms such as sneezing, itching, and runny nose caused by allergies.

Astelin Nasal Spray

Astelin nasal spray, an antihistamine medication, is a nasal spray used to alleviate the symptoms of seasonal allergic rhinitis and vasomotor rhinitis. Astelin contains the active ingredient azelastine hydrochloride, a white, crystalline powder with a bitter taste. Each metered spray delivers 137 mcg of azelastine hydrochloride.

The recommended dose for seasonal allergic rhinitis in adults and adolescents is one or two sprays per nostril twice daily.

For pediatric patients aged 5 to 11 years, the recommended dose is one spray per nostril twice daily.

For vasomotor rhinitis in patients aged 12 years or older, the recommended dose is two sprays per nostril twice daily.

Astelin should be primed before initial use and should not be sprayed into the eyes. It is important to follow the medication guide for comprehensive information on potential side effects and drug interactions.

Side Effects

It is important to understand the potential side effects of Astelin nasal spray. While it has been proven to relieve nasal congestion, which is a bothersome symptom for many allergy sufferers, Azelastine nasal spray may cause side effects. Therefore, it is crucial to be aware of these potential risks and consult with a healthcare professional if any side effects occur.

Understanding the Side Effects of Astelin Nasal Spray

The potential adverse reactions associated with the use of Astelin nasal spray encompass a range of symptoms and conditions that should be understood by patients and healthcare providers. Some common side effects of Astelin include:

  • A bitter taste in the mouth

  • Headache

  • Drowsiness

  • Nasal burning

  • Sore throat

  • Dry mouth

  • Sneezing

Some of the less common side effects of Astelin include:

  • Dizziness

  • Nosebleeds

  • Nausea

  • Red eyes

It is important for patients to be aware of these side effects and to report any concerning symptoms to their healthcare provider. Healthcare providers should also educate patients about the potential side effects and monitor them closely during treatment. By understanding the possible adverse reactions, patients and healthcare providers can work together to ensure the safe and effective use of Astelin nasal spray.

Azelastine Precautions

Azelastine nasal spray may result in various side effects that should be taken into consideration. While this medication is effective in relieving nasal symptoms of allergies, it can also cause some unwanted reactions.

It is important to note that serious side effects such as hives, difficulty breathing, and swelling of the face, lips, tongue, or throat may occur, although they are less common. This is a sign of an allergic reaction to the medication. If any of these severe side effects occur, it is crucial to seek medical attention immediately.

It is recommended to consult with a healthcare professional before using azelastine nasal spray to discuss potential side effects and determine if it is the right medication for you.

What Is the Active Ingredient in Astelin Nasal Spray?

Azelastine is the active ingredient in Astelin nasal spray, which is used to treat nasal symptoms of allergies. It is an antihistamine that helps prevent sneezing, itching, runny nose, and other allergy symptoms. Understanding the properties and effects of azelastine is important for healthcare professionals and patients who use Astelin nasal spray.

Azelastine hydrochloride is a white, crystalline powder with a bitter taste. It is sparingly soluble in water and slightly soluble in ethanol. Astelin contains 0.1% azelastine hydrochloride in an aqueous solution. Each metered spray delivers 137 mcg of azelastine hydrochloride.

This active ingredient works by blocking the effects of histamine, which is a substance produced by the body in response to allergens. By blocking histamine, azelastine helps to relieve symptoms such as sneezing, itching, and runny nose caused by allergies. It is important to follow the instructions provided by your healthcare provider and use Astelin nasal spray as directed for optimal results.

Before Using Azelastine Nasal Spray For the First Time

Before using azelastine nasal spray for the first time, it is important to familiarize yourself with the proper instructions and precautions to ensure safe and effective use. Azelastine nasal spray is an antihistamine spray that works by preventing the release of histamine, a substance in the body that causes allergic symptoms. It is available in generic form and contains 0.1% azelastine hydrochloride in an aqueous solution, delivering 137 mcg per spray.

To use azelastine nasal spray, first, prime the spray by pumping the bottle until a fine mist appears. This ensures that you receive the correct dose of medication. Then, blow your nose with a tissue to clear your nasal passages. Hold the bottle upright, insert the spray tip into one nostril with your head tilted forward, and close the other nostril with your finger. Breathe in gently through your nose while pressing down on the nasal spray pump to release the medication. Repeat these steps for the other nostril.

It is important to follow the instructions provided by your healthcare provider or the product label. Do not exceed the recommended dose or frequency of use. If you have any questions or concerns about using azelastine nasal spray, consult your healthcare provider for guidance.

What Happens if I Overdose?

After reviewing the instructions and precautions for using azelastine nasal spray, it is important to understand the potential consequences in the event of an overdose. An overdose occurs when an individual takes more medication than the prescribed amount, resulting in an excessive amount of the drug in the body.

In the case of azelastine nasal spray, an overdose may lead to various symptoms and side effects. These can include drowsiness, dizziness, headache, increased or irregular heartbeat, dry mouth, blurred vision, difficulty breathing, and even loss of consciousness. If you suspect an overdose of azelastine nasal spray, it is crucial to seek immediate medical attention.

Contact your healthcare provider, go to the nearest emergency room, or call your local poison control center for assistance. Provide them with information about the amount of medication taken, the time of ingestion, and any symptoms experienced. Prompt medical intervention can help prevent any serious complications and ensure appropriate treatment for an azelastine nasal spray overdose.

Patients should be instructed to keep Astelin Nasal Spray out of the reach of children and to avoid spraying it into their eyes. If a child accidentally ingests Astelin Nasal Spray, seek immediate medical help or call a poison control center.

What Other Drugs Will Affect Astelin?

Concurrent use of other medications with Astelin may result in potential drug interactions. It is important to be aware of these interactions to ensure the safe and effective use of Astelin. A primary concern is the combination of Astelin and central nervous system depressants, such as alcohol and sedatives. When used together, these substances can cause reductions in alertness and impairment of central nervous system performance. Therefore, it is recommended to avoid concurrent use of Astelin with alcohol or other central nervous system depressants.

Drug Interactions

Astelin is metabolized by the cytochrome P450 enzyme system, although the specific P450 isoforms responsible for its biotransformation have not been identified. Co-administration of azelastine with erythromycin, cimetidine, or theophylline does not result in significant pharmacokinetic interactions.

Co-administration of erythromycin with Astelin may increase the concentrations of Astelin in the body. Additionally, theophylline, a medication used to treat respiratory conditions, does not result in significant pharmacokinetic interactions when taken with Astelin.

It is important to inform your healthcare provider about all medications you are taking, including prescription, over-the-counter, and herbal supplements, to avoid any potential interactions with Astelin. Your healthcare provider can determine if any adjustments to your medication regimen are necessary to ensure the safe and effective use of Astelin.

Dosage Forms And Strengths

Astelin is available in different dosage forms and strengths to accommodate the needs of patients requiring treatment for nasal symptoms of allergies. It is primarily available as a nasal spray, containing 0.1% azelastine hydrochloride in an aqueous solution. Each metered spray delivers 137 mcg of azelastine hydrochloride.

The recommended dosage of Astelin varies depending on the age and condition being treated. For adults and adolescents with seasonal allergic rhinitis, the recommended dose is one or two sprays per nostril, twice daily. Pediatric patients aged 5 to 11 years should use one spray per nostril, twice daily.

For the treatment of vasomotor rhinitis in patients aged 12 years or older, the recommended dose is two sprays per nostril, twice daily.

It is important to prime the Astelin nasal spray before initial use and to reprime it if it has not been used for 3 or more days. Avoid spraying Astelin into the eyes.

Additional Information

In addition to the dosage forms and strengths of azelastine nasal spray, there are several important points to consider. These include what to do if a dose is missed, the use of azelastine for seasonal allergic rhinitis, potential interactions with other medications, and how certain medical conditions may affect the use of azelastine. It is important to be aware of these points to ensure the safe and effective use of the medication.

What Happens if I Miss a Dose?

If a dose of Astelin is missed, it is important to take the missed dose as soon as possible. However, if it is almost time for the next dose, skip the missed dose and continue with the regular dosing schedule. Do not double the dose to make up for the missed one.

It is crucial to follow the prescribed dosing instructions and not exceed the recommended dosage. Taking more than the prescribed amount may increase the risk of side effects. If you have any concerns or questions about missed doses or the proper use of Astelin, it is recommended to consult with a healthcare professional or pharmacist who can provide guidance and answer any specific questions you may have.

Other Medical Problems

Other medical conditions should be taken into consideration when using Astelin, an antihistamine nasal spray used to treat nasal symptoms of allergies. It is important to consult with a healthcare professional before using Astelin if you have any of the following medical problems: asthma, nasal ulcers or have had nasal surgery, open sores or injuries in the nose, or an untreated infection in the nose or sinuses.

Additionally, individuals with a history of allergic reactions to azelastine or other antihistamines should avoid using Astelin.

Patients with liver or kidney disease may require dosage adjustments or special monitoring while using this medication. It is crucial to disclose all relevant medical information to your healthcare provider to ensure safe and effective use of Astelin.

Proper Use

Keep Spray Out of Eyes

To ensure the proper use of Astelin Nasal Spray and prevent potential eye irritation, it is essential to take precautions and keep the spray out of the eyes. Astelin is intended for use only as a nasal spray, despite its ability to help manage itchy, watery eyes. Using the nasal spray directly on the eyes results in irritation and discomfort. The best way to use a nasal spray is to blow your nose first and insert the nozzle just inside the rounded part of your nostril. Keep a tissue nearby. If a small portion drips out, this is okay.

It is crucial to avoid spraying the medication into the eyes. Patients should be instructed to keep the spray out of the reach of children and seek immediate medical help if a child accidentally ingests it.

Astelin Nasal Spray Two Sprays Per Nostril Twice Daily For Patients 12 Years And Older

To properly use Astelin Nasal Spray, it is recommended to administer two sprays per nostril twice daily for patients 12 years of age and older. This dosage regimen is effective in treating seasonal allergic rhinitis and vasomotor rhinitis symptoms such as sneezing, itching, and runny nose caused by allergies.

Astelin can be used in patients as young as 5 years old at a dose of one spray twice daily for allergy symptoms.

Before initial use and if not used for 3 or more days, the nasal spray should be primed. It is important to avoid spraying Astelin into the eyes and to keep it out of the reach of children. If a child accidentally ingests Astelin Nasal Spray, seek immediate medical help or call a poison control center. By following the recommended dosage and administration instructions, individuals can effectively manage their nasal allergy symptoms and improve their overall quality of life.

Frequently Asked Questions

Can I Use Azelastine Nasal Spray While Pregnant or Breastfeeding?

Azelastine nasal spray should be used with caution in pregnant women. It is recommended to consult with a healthcare professional before using this medication during pregnancy or while breastfeeding to assess potential risks and benefits.

How Long Does It Take for Azelastine Nasal Spray to Start Working?

The onset of action for Azelastine nasal spray can vary, but it typically starts working within 15-30 minutes after administration. However, individual response may vary. It is best to follow the recommended dosing instructions and consult with a healthcare professional for personalized advice.

Can Azelastine Nasal Spray Be Used in Children Younger Than 5 Years Old?

Azelastine nasal spray is indicated for use in patients as young as 5 years old. However, it is important to consult with a healthcare professional for appropriate dosage and administration in children of this age group.

Can I Use Azelastine Nasal Spray if I Have a History of High Blood Pressure?

Azelastine nasal spray should be used with caution if you have a history of high blood pressure. Consult your healthcare provider to determine if it is safe for you to use this medication.

Is Azelastine Nasal Spray Addictive?

No, Azelastine nasal spray is not addictive. It is an antihistamine nasal spray used to treat nasal symptoms of allergies and does not have addictive properties. However, it should be used as directed by a healthcare professional.

Finding Quality Azelastine at Heavily Discounted Prices

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The content on this page is for informational and educational purposes only and does not constitute professional medical advice. Patients should not use the information presented on this page for diagnosing a health-related issue or disease. Before taking any medication or supplements, patients should always consult a physician or qualified healthcare professional for medical advice or information about whether a drug is safe, appropriate or effective.